Here we report within the success of the strategy, including biochemical, biophysical, and cellular evidence of the desired irreversible covalent inhibition
Here we report within the success of the strategy, including biochemical, biophysical, and cellular evidence of the desired irreversible covalent inhibition. higher dehydration penalty could also be expected for secondary amides versus tertiary ones upon complex formation. Open in a separate windowpane Fig. 2. Rendering from the 2 2.70-? X-ray crystal structure (5TER) of 1 […]